Explore Exerkines

Browse 35 exercise-induced signaling molecules by therapeutic domain and translational tier

Translational Readiness Tiers

Each exerkine is assigned a tier reflecting its stage along the bench-to-bedside pipeline:

1 Clinically Validated — Approved therapeutics or advanced clinical trials with regulatory milestones
2 Clinical Trials — Active or completed human trials; strong mechanistic and preclinical evidence
3 Preclinical Promise — Robust in vivo data in animal models; clinical translation not yet initiated
4 Emerging Targets — Early-stage research with suggestive but limited evidence; further validation required
Therapeutic Domains & Evidence Symbols

The table scores each exerkine across six therapeutic domains based on the strength and breadth of published evidence:

CV
Cardiovascular (heart failure, atherosclerosis, hypertension)
Met
Metabolic (obesity, type 2 diabetes, insulin resistance)
Neuro
Neurological (neurodegeneration, cognitive decline, depression)
MSK
Musculoskeletal (sarcopenia, bone loss, joint health)
Inflam
Anti-inflammatory (chronic inflammation, immune modulation)
Onco
Oncology (tumor suppression, cancer risk reduction)

Evidence symbols

●● Primary domain (strongest evidence) Established evidence Preliminary evidence ○* Dual / complex role ●(t) Target for inhibition Not reported
Exerkine Tier Source Tissue CV Met Neuro MSK Inflam Onco
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